Heterologous Modulation of Androgen Receptor Nucleo-Cytoplasmic Shuttling by Melatonin: A Novel Mode of Regulating Androgen Sensitivity
Melatonin, the hormone secreted nocturnally from the pineal gland, is an androgen protagonist in vivo. Its effects are mostly demonstrable under conditions of low circulating androgen levels (e.g., during pubertal development, under conditions of chemical or surgical castration or androgen ablation therapy). The prostate gland is an androgen dependent organ that responds to melatonin in vivo. Benign and cancer prostate cells provide suitable systems for exploring androgen-melatonin interactions in vitro.
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